Virological failure to raltegravir in Spain: incidence, prevalence and clinical consequences


Por: Santos, JR, Blanco, JL, Masia, M, Gutierrez, F, Perez-Elias, MJ, Iribarren, JA, Force, L, Antela, A, Knobel, H, Salavert, M, De Quiros, JCLB, Pino, M, Paredes, R and Clotet, B

Publicada: 1 nov 2015
Resumen:
Objectives: The objective of this study was to evaluate the incidence, prevalence and clinical consequences of virological failure (VF) to raltegravir-based regimens in Spain. Methods: A multicentre, retrospective, observational study was performed in 10 tertiary hospitals (January 2006 to June 2013). The study included HIV-1-infected patients with loss of virological suppression (LVS; two consecutive HIV-1 RNA >= 50 copies/mL) while receiving raltegravir. VF and low-level viraemia (LLV) were defined as two consecutive HIV-1 RNA = 200 copies/mL and 50 to <200 copies/mL, respectively. Integrase strand-transfer inhibitor resistance was investigated at LVS. During the 48 weeks following LVS, recorded data included clinical characteristics, treatment discontinuations, AIDS-associated events and deaths. Effectiveness of therapy following LVS was evaluated by ITT and PP. Multivariate regression was used to assess predictors of efficacy. Results: Of the 15009 HIV-infected patients in participating centres, 2782 (18.5%) had received raltegravir-based regimens. Of those, 192 (6.9%), 125 (4.5%) and 67 (2.4%) experienced LVS, VF and LLV, respectively. The incidence of VF was 1.8 (95% CI, 1.5-2.1) per 100 patients/year. The prevalence of VF was 4.5% (95% CI, 3.8%-5.3%). Integrase-associated mutations were found in 78.8% of patients with integrase genotyping results available. High-level resistance to dolutegravir was not observed. Salvage therapy failed in 34.1% of patients; progression to AIDS/death occurred in 8.3% during the first year following LVS. The latter was associated with intravenous drug use, time on raltegravir and lower CD4+ count nadir in patients who started raltegravir-based treatments as salvage regimens. Conclusions: VF with raltegravir is infrequent, but often associated with major clinical complications in treatment-experienced patients.

Filiaciones:
:
 Hosp Univ Germans Trias I Pujol, Fundacio Lluita SIDA, Barcelona 08916, Spain

 Univ Autonoma Barcelona, E-08193 Barcelona, Spain

Blanco, JL:
 Univ Barcelona, Hosp Clin Barcelona, IDIBAPS, Barcelona, Spain

Masia, M:
 Elche Univ Gen Hosp, Infect Dis Unit, Elche, Spain

 Miguel Hernandez Univ, Elche, Spain

Gutierrez, F:
 Elche Univ Gen Hosp, Infect Dis Unit, Elche, Spain

 Miguel Hernandez Univ, Elche, Spain

Perez-Elias, MJ:
 Hosp Ramon & Cajal, IRYCIS, Infect Dis Unit, E-28034 Madrid, Spain

Iribarren, JA:
 Donostia Univ Hosp, Infect Dis Unit, San Sebastian, Spain

Force, L:
 Mataro Hosp, Infect Dis Unit, Mataro, Spain

Antela, A:
 Univ Hosp, Infect Dis Unit, Santiago De Compostela, Spain

Knobel, H:
 IMIM Hosp Mar Res Inst, Hosp Mar, Infect Dis Serv, Barcelona, Spain

Salavert, M:
 La Fe Univ, Infect Dis Unit, Valencia, Spain

 Polytech Hosp, Valencia, Spain

De Quiros, JCLB:
 Gregorio Maranon Univ Hosp, Infect Dis Unit, Madrid, Spain

Pino, M:
 IrsiCaixa AIDS Res Inst, Barcelona, Spain

:
 Hosp Univ Germans Trias I Pujol, Fundacio Lluita SIDA, Barcelona 08916, Spain

 IrsiCaixa AIDS Res Inst, Barcelona, Spain

 Univ Vic Univ Cent Catalunya, Vic, Spain

:
 Hosp Univ Germans Trias I Pujol, Fundacio Lluita SIDA, Barcelona 08916, Spain

 Univ Autonoma Barcelona, E-08193 Barcelona, Spain

 IrsiCaixa AIDS Res Inst, Barcelona, Spain

 Univ Vic Univ Cent Catalunya, Vic, Spain
ISSN: 03057453





Journal of Antimicrobial Chemotherapy
Editorial
Oxford University Press, GREAT CLARENDON ST, OXFORD OX2 6DP, ENGLAND, Reino Unido
Tipo de documento: Article
Volumen: 70 Número: 11
Páginas: 3087-3095
WOS Id: 000368245500022
ID de PubMed: 26490727

MÉTRICAS